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Search Results for " adenylate cyclase "

46

抑制剂 & 化合物

4

天然产物

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Cat. No.	Product Name	Target	Signaling Pathways
T15658	KH7	cAMP; AChR	GPCR/G Protein; Neuroscience
	KH7 是腺苷酸环化酶 (sAC) 特异性的可溶性抑制剂，也是一种 cAMP 抑制剂。它对重组纯化的人类 sACt 蛋白和细胞试验中异源表达的 sACt 的 IC50 为 3 到 10 μM 之间。
T16938	ST034307	Adenylyl cyclase	Neuroscience
	ST034307 是一种选择性 adenylyl cyclase 1抑制剂，IC50值为 2.3 μM。
T0322	Fipexide	Dopamine Receptor; AChR	GPCR/G Protein; Neuroscience
	Fipexide 是对氯苯乙酸衍生物，是哌嗪化学类的精神活性药物，作为促智药物，有用于老年痴呆的研究潜力。它可降低了纹状体腺苷酸环化酶的活性，通过多巴胺能神经传递对认知表现出积极的作用。
T10066	2',5'-Dideoxyadenosine	Adenylyl cyclase; Adrenergic Receptor; AChR	GPCR/G Protein; Neuroscience
	2',5'-Dideoxyadenosine 是一种非竞争性腺苷酸环化酶抑制剂，通过结合 P 位点，IC50为 3 µM。它是核苷类似物，在心脏中发挥强大的抗肾上腺素作用。
T60003	AC1-IN-1	Adenylyl cyclase	Neuroscience
	AC1-IN-1 是 1 型腺苷酸环化酶的选择性抑制剂（AC1，IC50 = 0.54 µM）。
T16275	NB001 HTS 09836	Adenylyl cyclase	Neuroscience
	NB001 (HTS 09836) 是腺苷酸环化酶 1 的抑制剂，对神经和非神经疼痛有作用。
T8702	SKF-83566	Dopamine Receptor; 5-HT Receptor; AChR	GPCR/G Protein; Neuroscience
	SKF-83566 是一种具有血脑渗透性和口服活性的 D1 样多巴胺受体拮抗剂和一种较弱的竞争性 5-HT2 受体拮抗剂，Ki 为 11 nM。它是竞争性多巴胺转运蛋白抑制剂，可用于研究帕金森氏症和对尼古丁渴望的缓解的相关研究。
T0830	Bithionol 硫双二氯酚,Actamer,硫氯酚	cAMP; Parasite	GPCR/G Protein; Microbiology/Virology
	Bithionol (Actamer) 是一种抗寄生虫药物，对若干癌细胞有抑制作用。
T2172	SQ22536 9-(tetrahydrofuran-2-yl)-9h-purin-6-amine,SQ 22536	AChR	Neuroscience
	SQ22536 (9-(tetrahydrofuran-2-yl)-9h-purin-6-amine) 是一种腺苷酸环化酶抑制剂。
T80069	PACAP (6-27) (human, ovine, rat) Pituitary adenylate cyclase-activating peptide (6-27)
	PACAP (6-27) (human, ovine, rat) 是一种对PACAP受体具有拮抗作用的化合物，可以抑制犬肾上腺对外源性VIP的反应。此化合物在心血管疾病和神经系统疾病研究中展现出应用潜力。
TP1878	PACAP (1-38), human, ovine, rat Pituitary Adenylate Cyclase Activating Polypeptide 38,腺苷酸环化酶激活肽-38(抗原),PACAP 1-38	PACAP	GPCR/G Protein
	PACAP (1-38), human, ovine, rat (Pituitary Adenylate Cyclase Activating Polypeptide 38) 是含有 38 个氨基酸残基的神经肽。它能够结合 PACAP I 型受体(IC50:4 nM)、PACAP II 型受体 VIP1(IC50:2 nM)、PACAP II 型受体 VIP2(IC50:1 nM)。
TP1054	PACAP (1-38), human, ovine, rat TFA Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA)
	PACAP (1-38), a novel neuropeptide isolated from the bovine hypothalamus is more active than vasoactive intestinal peptide (VIP) in stimulating adenylate cyclase (EC50=7 nM). PACAP 1-38 (10-9 M) increased substance P (SP), gastrin releasing peptide (GRP),
T11918	Lysipressin Lysine vasopressin,[Lys8]-Vasopressin,赖氨加压素	Others	Others
	Lysipressin ([Lys8]-Vasopressin) 是一种抗利尿激素，从猪身上发现，能够诱发兔膀胱平滑肌的收缩，激活腺苷酸环化酶。
T14880	CB-7921220 6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid,6-(4-Aminostyryl)picolinic acid,6-[(E)-2-(4-aminophenyl)ethenyl]pyridine-2-carboxylic acid	AChR	Neuroscience
	CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid)是一种腺苷酸环化酶的抑制剂。
T29652	9-Cyclopentyladenine NSC19486,NSC 19486,9CPAde,9-CP-Ade,9 CP Ade,NSC-19486	AChR	Neuroscience
	9-Cyclopentyladenine (NSC-19486) 是一种腺苷酸环化酶抑制剂，可阻断细胞形态分化和特定信号分子磷酸化。
T23588	9-CP-Ade Mesylate 9-Cyclopentyladenine monomethanesulfonate,9 CP Ade Mesylate,9CPAde Mesylate	AChR	Neuroscience
	9-CP-Ade Mesylate (9 CP Ade Mesylate)是一种具有细胞渗透性的、稳定性和非竞争性的腺苷酸环化酶 (adenylate cyclase) 抑制剂。
T22489	2'-MeCCPA 2-Chloro-N-cyclopentyl-2′-C-methyladenosine	HCV Protease; Adenosine Receptor	GPCR/G Protein; Microbiology/Virology; Neuroscience; Proteases/Proteasome
	2'-MeCCPA 是一种具有有效性和高选择性的 A1 腺苷受体 (A1AR) 激动剂，对 AR 的 K 值为 1.8 nM。2'-MeCCPA 抑制毛喉素刺激的腺苷酸环化酶活性，IC值为13.1 nM。2'-MeCCPA 具有镇痛活性，可用于研究 HCV 。
T11918L	Lysipressin acetate(50-57-7(fb_acetate)) Lysine vasopressin acetate,[Lys8]-Vasopressin acetate	Others	Others
	Lysipressin acetate(50-57-7(fb_acetate)) ([Lys8]-Vasopressin acetate) 诱导兔膀胱平滑肌收缩，激活腺苷酸环化酶。 Lysipressin 是一种抗利尿激素，已在猪和一些有袋动物家族中发现。
T78105	PAC1R antagonist 1	PACAP	GPCR/G Protein
	PAC1R antagonist 1为一种具有口服活性的 PAC1 受体拮抗剂，可抑制由垂体腺苷酸环化酶激活多肽（PACAP）及神经损伤所诱导的异常性疼痛，可用于研究肿瘤和与免疫相关的疾病。
TP1878L	PACAP 1-38 acetate	PACAP	GPCR/G Protein
	PACAP 1-38 acetate 是一种垂体腺苷酸环化酶激活多肽 (PACAP) 类似物。它与 PACAP I 型受体 (IC50 = 4 nM) 和 PACAP II 型 VIP2 受体 (IC50 = 1 nM) 结合，但不与 PACAP II 型 VIP1 受体结合。
TP1844L	Small Cardioactive Peptide B SCPB acetate Small Cardioactive Peptide B SCPB acetate(84746-43-0 free base)	Others	Others
	Small Cardioactive Peptide B SCPB acetate (Small Cardioactive Peptide B SCPB acetate (84746-43-0 free base)) 是一种神经活性肽，可刺激心脏和鳃组织颗粒部分的腺苷酸环化酶活性，EC50 分别为 0.1 和 1.0 μM。
T4436	RO1138452 CAY10441	Others; Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation; Others
	RO1138452 (CAY10441) 是一种选择性和可口服的前列环素受体拮抗剂，pKi 为8.3。它拮抗卡前列环素诱导的人神经母细胞瘤腺苷酸环化酶的激活，以剂量依赖性方式阻断环 AMP 积累，具有镇痛活性。
T1139	Salbutamol Albuterol,沙丁胺醇,AH-3365	Adrenergic Receptor	GPCR/G Protein; Neuroscience
	Salbutamol (Albuterol) 是短效的 β2 肾上腺素受体激动剂，用于哮喘和慢性阻塞性肺疾病(COPD) 引发的支气管痉挛的研究。
T37477	L-858,051 (hydrochloride)
	L-858,051 is a water-soluble analog of forskolin , a cell-permeant activator of adenylate cyclase. L-858,051 activates adenylate cyclase (EC50 = 3 μM), inhibits glucose transport, and blocks cytochalasin B binding in rat adipocyte membranes. L-858,051 is used to activate adenylate cyclase and initiate signaling through elevated cAMP synthesis in a variety of cell types in culture.
T24365	L 858051 7B-Forskolin,L858051,Dmpb-forskolin,L-858051
	L 858051 activates adenylate cyclase. It also inhibits glucose transport in rat adipocytes.
T31751	Fce 21258 Ddh-carbo pgl2
	Fce 21258 is used to stimulate the adenylate cyclase of synovial fluid macrophages.
T27057	CP 154,526 CP-154,526,CP154,526
	CP 154,526 is a selective CRF1 receptor antagonist (Ki = 2.7 nM). CP 154,526 blocks CRF-induced activation of adenylate cyclase and the HPA axis.
T70581	CY208-243 Mandelate
	CY208-243 is a D1 agonist. CY208-243 attenuates the pattern electroretinogram to low spatial frequency stimuli in the monkey. CY208-243 stimulates adenylate cyclase in rat striatal homogenates with an EC50 of 125 nM. CY208,243 was superior in improving the strength of neuronal outcome sensitivity to the working memory-related choice behavior in the T-maze.
T36009	Guanylyl Imidodiphosphate (lithium salt)
	Guanylyl Imidodiphosphate (lithium salt) 是一种 GTP 类似物，不可水解，可增加腺苷酸环化酶 (adenylate cyclase) 活性。
T26536	AC-178335 AC 178335,AC178335
	AC-178335 is a pure somatostatin (SRIF) antagonist with an affinity constant (Ki) of 172 +/- 12 nM. AC-178335 blocks SRIF inhibition of adenylate cyclase in vitro (IC50 = 5.1 +/- 1.4 microM). It induces GH release when given alone (50 micrograms intraveno
TP1844	Small Cardioactive Peptide B (SCPB) Small Cardioactive Peptide B SCPB
	Small Cardioactive Peptide B (SCPB), a neurally active peptide, stimulates adenylate cyclase activity in particulate fractions of both heart and gill tissues with EC50s of 0.1 and 1.0 μM, respectively.
T82306	Glucagon (22-29)
	Glucagon (22-29) 作为Glucagon (19–29)的部分激动剂，能特异性抑制肝质膜 Ca2+泵，其作用机制与腺苷酸环化酶激活无关。
T21803	Guanylyl Imidodiphosphate
	Guanylyl Imidodiphosphate (Guanosine 5'-[β,γ-imido]triphosphate) trisodium 是一种不可水解的 GTP 类似物，是ADP-核糖基化因子 (ARF) 激活剂和腺苷酸环化酶 (adenylate cyclase) 的有效刺激物。Guanylyl Imidodiphosphate trisodium 可用于蛋白质合成研究。
T38055	Salvinorin A Propionate
	Salvinorin A propionate is a selective partial agonist at κ1-opioid receptors (KOR) with a Ki value of 32.6 nM. It inhibits adenylate cyclase (EC50 = 4.7 nM) in HEK293 cells transfected with human KOR. It is selective for KORs over μ, δ, and ORL-1 opioid receptors and has no effect at serotonin, dopamine, muscarinic, or adrenergic receptors. In mice, salvinorin A propionate (13 μg, i.c.v.) reduces nociceptive responses in a radiant heat tail-flick assay, though not as potently as salvinorin A .
TP1722	PACAP (6-38), human, ovine, rat
	PACAP (6-38), human, ovine, rat is a potent antagonist of PACAP 38. PACAP (6-38) is much more potent and selective than PACAP (6-27) in the inhibition of PACAP-27-stimulated pituitary adenylate cyclase.
T36072	Skyrin Endothianin,Rhodophyscin
	Skyrin is a fungal metabolite characterized by a bisanthraquinone structure. It interferes with glucagon signaling through adenylate cyclase without binding to the glucagon receptor. At 10 μM, skyrin reduces both glucagon-stimulated cAMP production and glycogenolysis. It does not interfere with epinephrine or glucagon-like peptide 1 effects on these parameters.[1] Reference：[1]. Parker, J.C., McPherson, R.K., Andrews, K.M., et al. Effects of skyrin, a receptor-selective glucagon antagonist, in r...
T76363	[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
	[Tyr22]CalcitoninGene Related Peptide, (22-37), rat 是一种大鼠降钙素基因相关肽 (CGRP) 的 22-37 片段，靶向CGRP 受体和腺苷酸环化酶。降钙素 (calcitonin) 主要由甲状腺 C 细胞产生，而 CGRP 则分泌并储存在神经系统中。
T37435	PACAP-related Peptide (rat) (trifluoroacetate salt)	PACAP	GPCR/G Protein
	PACAP-related peptide (PRP) is an endogenous 29-amino acid peptide that belongs to the secretin/glucagon superfamily of peptides, which includes secretin , glucagon , glucagon-like peptide-1 , GLP-2 , and pituitary adenylate cyclase-activating polypeptide . It is expressed in rat hypothalamus as well as within the nerves of the median eminence, the anterior pituitary, bed nucleus of the stria terminalis, cerebellum, cerebral cortex, and amygdala. PRP is also expressed in vaginal, uterine cervica...
T36428	PACAP-related Peptide (human) (trifluoroacetate salt)	PACAP	GPCR/G Protein
	PACAP-related peptide (PRP) is an endogenous 29-amino acid peptide that belongs to the secretin/glucagon superfamily of peptides, which includes secretin , glucagon , glucagon-like peptide-1 , GLP-2 , and pituitary adenylate cyclase-activating polypeptide . It is expressed in normal human pancreas and adrenal gland tissue and in some tumors that produce vasoactive intestinal peptide (VIP). PRP (1-29) is secreted by CHO-K1 cells that express human recombinant preproPACAP.
T36236	5-cis Carbaprostacyclin
	5-cis Carbaprostacyclin is a stable analog of PGI2 and an isomer of carbaprostacyclin. It is a weak inhibitor of human platelet aggregation with an IC50 of 2.8 μM compared to 0.3 μM for carbaprostacyclin. 5-cis Carbaprostacyclin is a much weaker effector of rabbit mesenteric artery relaxation with an EC50 of 104 μM compared to 5.9 μM for carbaprostacyclin. It even antagonizes the adenylate cyclase activation induced by carbaprostacyclin.
T36239	6β-Prostaglandin I1 6β-Prostaglandin I1
	6β-PGI1 is a stable PGI2 analog resistant to hydrolysis in aqueous solutions. 6β-PGI1 has a much longer half-life than PGI2, but a greatly reduced molar potency for receptor mediated function. 6β-PGI1 has a Kact for adenylate cyclase in NCB-20 cells of 4.2 μM compared with 18 nM for PGI2. The potency for vasodilation and inhibition of platelet aggregation is about 1% of PGI2.
T36427	PACAP (6-27) (human, chicken, mouse, ovine, porcine, rat) (trifluoroacetate salt)	PACAP	GPCR/G Protein
	Pituitary adenylate cyclase-activating peptide (PACAP) (6-27) is a PACAP receptor antagonist with IC50 values of 1,500, 600, and 300 nM, respectively, for rat PAC1, rat VPAC1, and human VPAC2 recombinant receptors expressed in CHO cells. It binds to PACAP receptors on SH-SY5Y and SK-N-MC human neuroblastoma and T47D human breast cancer cells (IC50s = 24.5, 106, and 105 nM, respectively) and inhibits cAMP accumulation induced by PACAP (1-38) (Kis = 457, 102, and 283 nM, respectively, in SH-SY5Y, ...
T70865	BMY-42393
	BMY-42393 is orally active and selective platelet aggregation inhibitor. BMY-42393 is also a prostacyclin partial agonist that inhibited ADP, collagen and thrombin-induced platelet aggregation (IC50 range 0.3 - 2.0 microM). BMY-42393 stimulated platelet adenylate cyclase activity (EC50 = 25 nM). Platelets treated with BMY 42393 showed an elevation of cAMP levels and activation of cAMP-dependent protein kinase. BMY 42393 also inhibited thrombin-induced elevation of intracellular free calcium. B...
T36775	13,14-dihydro Prostaglandin E1 13,14-dihydro Prostaglandin E1
	13,14-dihydro Prostaglandin E1 (13,14-dihydro PGE1) is a biologically active metabolite of PGE1 with comparable potency to the parent compound. It is an inhibitor of ADP-induced platelet aggregation in human PRP and washed platelets with IC50 values of 31 and 21 nM, respectively. 13,14-dihydro PGE1 is a slightly more potent inhibitor of ADP-induced human platelet aggregation than PGE1 which has an IC50 value of 40 nM. Also, 13,14-dihydro PGE1 was shown to activate adenylate cyclase in NCB-20 hyb...
T76042	Angiopeptin TFA
	Angiopeptin TFA，一种生长抑素的环状八肽类似物，作为sst2/sst5受体部分激动剂，其IC50值为0.26 nM和6.92 nM。该化合物能够抑制生长激素释放及IGF-1(胰岛素样生长因子-1)的产生，同时抑制腺苷酸环化酶活性或刺激细胞外酸化。Angiopeptin TFA在冠状动脉粥样硬化的研究中显示出潜力。
T36720	Deacetylforskolin
	Deacetylforskolin is a diterpene and a derivative of forskolin that has been found inC. forskohliiand has diverse biological activities.1,2,3,4It activates rat adipocyte adenylyl cyclase (IC50= 20 μM) and inhibits glucose transport in rat adipocyte plasma membranes.2Deactylforskolin (30-1,000 μg/kg) reduces blood pressure in spontaneously hypertensive rats.3It also attenuates hypercapnia-induced impairments in the passive avoidance response in mice.4 1.Gabetta, B., Zini, G., and Danieli, B.Minor...

化合物

Cat.No: T15658

Target: cAMP, AChR

Cat.No: T16938

Target: Adenylyl cyclase

Cat.No: T0322

Target: Dopamine Receptor, AChR

2',5'-Dideoxyadenosine

Cat.No: T10066

Target: Adenylyl cyclase, Adrenergic Receptor, AChR

Cat.No: T60003

Target: Adenylyl cyclase

Cat.No: T16275

Synonym: HTS 09836

Target: Adenylyl cyclase

Cat.No: T8702

Target: Dopamine Receptor, 5-HT Receptor, AChR

Cat.No: T0830

Synonym: 硫双二氯酚,Actamer,硫氯酚

Target: cAMP, Parasite

Cat.No: T2172

Synonym: 9-(tetrahydrofuran-2-yl)-9h-purin-6-amine,SQ 22536

Target: AChR

PACAP (6-27) (human, ovine, rat)

Cat.No: T80069

Synonym: Pituitary adenylate cyclase-activating peptide (6-27)

PACAP (1-38), human, ovine, rat

Cat.No: TP1878

Synonym: Pituitary Adenylate Cyclase Activating Polypeptide 38,腺苷酸环化酶激活肽-38(抗原),PACAP 1-38

Target: PACAP

PACAP (1-38), human, ovine, rat TFA

Cat.No: TP1054

Synonym: Pituitary Adenylate Cyclase Activating Polypeptide 38 (TFA)

Cat.No: T11918

Synonym: Lysine vasopressin,[Lys8]-Vasopressin,赖氨加压素

Target: Others

Cat.No: T14880

Synonym: 6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid,6-(4-Aminostyryl)picolinic acid,6-[(E)-2-(4-aminophenyl)ethenyl]pyridine-2-carboxylic acid

Target: AChR

9-Cyclopentyladenine

Cat.No: T29652

Synonym: NSC19486,NSC 19486,9CPAde,9-CP-Ade,9 CP Ade,NSC-19486

Target: AChR

9-CP-Ade Mesylate

Cat.No: T23588

Synonym: 9-Cyclopentyladenine monomethanesulfonate,9 CP Ade Mesylate,9CPAde Mesylate

Target: AChR

Cat.No: T22489

Synonym: 2-Chloro-N-cyclopentyl-2′-C-methyladenosine

Target: HCV Protease, Adenosine Receptor

Lysipressin acetate(50-57-7(fb_acetate))

Cat.No: T11918L

Synonym: Lysine vasopressin acetate,[Lys8]-Vasopressin acetate

Target: Others

PAC1R antagonist 1

Cat.No: T78105

Target: PACAP

PACAP 1-38 acetate

Cat.No: TP1878L

Target: PACAP

Small Cardioactive Peptide B SCPB acetate

Cat.No: TP1844L

Synonym: Small Cardioactive Peptide B SCPB acetate(84746-43-0 free base)

Target: Others

Cat.No: T4436

Synonym: CAY10441

Target: Others, Prostaglandin Receptor

Cat.No: T1139

Synonym: Albuterol,沙丁胺醇,AH-3365

Target: Adrenergic Receptor

L-858,051 (hydrochloride)

Cat.No: T37477

Cat.No: T24365

Synonym: 7B-Forskolin,L858051,Dmpb-forskolin,L-858051

Cat.No: T31751

Synonym: Ddh-carbo pgl2

Cat.No: T27057

Synonym: CP-154,526,CP154,526

CY208-243 Mandelate

Cat.No: T70581

Guanylyl Imidodiphosphate (lithium salt)

Cat.No: T36009

Cat.No: T26536

Synonym: AC 178335,AC178335

Small Cardioactive Peptide B (SCPB)

Cat.No: TP1844

Synonym: Small Cardioactive Peptide B SCPB

Glucagon (22-29)

Cat.No: T82306

Guanylyl Imidodiphosphate

Cat.No: T21803

Salvinorin A Propionate

Cat.No: T38055

PACAP (6-38), human, ovine, rat

Cat.No: TP1722

Cat.No: T36072

Synonym: Endothianin,Rhodophyscin

[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat

Cat.No: T76363

PACAP-related Peptide (rat) (trifluoroacetate salt)

Cat.No: T37435

Target: PACAP

PACAP-related Peptide (human) (trifluoroacetate salt)

Cat.No: T36428

Target: PACAP

5-cis Carbaprostacyclin

Cat.No: T36236

6β-Prostaglandin I1

Cat.No: T36239

Synonym: 6β-Prostaglandin I1

PACAP (6-27) (human, chicken, mouse, ovine, porcine, rat) (trifluoroacetate salt)

Cat.No: T36427

Target: PACAP

Cat.No: T70865

13,14-dihydro Prostaglandin E1

Cat.No: T36775

Synonym: 13,14-dihydro Prostaglandin E1

Angiopeptin TFA

Cat.No: T76042

Deacetylforskolin

Cat.No: T36720

Cat. No.	Product Name	Target	Signaling Pathways
T2939	Forskolin 毛喉素,Coleonol,Colforsin	FXR; Adenylyl cyclase; AChR; Autophagy	Autophagy; Metabolism; Neuroscience
	Forskolin (Coleonol) 属于天然产物，是一种腺苷酸环化酶激活剂 (EC50=0.5 μM)。Forskolin 可以增加 cAMP 水平，可以激活 PXR 和 FXR，也可以诱导细胞自噬。Forskolin 对心脏产生正性肌力作用，具有血小板抗凝集和降压作用。
T1723	Adenosine 5'-diphosphate 腺苷5'-二磷酸,Adenosine diphosphate,adenosine pyrophosphate,ADP	Endogenous Metabolite	Metabolism
	Adenosine 5'-diphosphate (ADP) 是一种嘌呤核糖核苷5'-二磷酸，是 ATP 在 ATP 酶作用下去磷酸化的产物。Adenosine 5'-diphosphate (adenosine pyrophosphate) 可诱导人血小板聚集并通过作用于P2T-嘌呤受体抑制受刺激的腺苷酸环化酶。
T1626	Prostaglandin E1 前列地尔,PGE1,列腺素E1,Alprostadil	Endogenous Metabolite; Prostaglandin Receptor	GPCR/G Protein; Immunology/Inflammation; Metabolism
	Prostaglandin E1 (Alprostadil) 是一种前列腺素受体配体，对小鼠 EP1、EP2、EP3、EP4和 IP 的 Ki 值分别为 36、10、1.1、2.1 和 33 nM。它诱导血管舒张并抑制血小板聚集，可作为血管扩张剂用于外周血管疾病的研究。
T16332	NKH477 Colforsin dapropate hydrochloride	NMDAR	Neuroscience
	NKH477 is a novel water-soluble forskolin derivative that improves cardiac failure mainly through its beneficial effects on diastolic cardiac function. NKH477 shows an antiproliferative effect in vivo with an altered cytokine profile to inhibit the acute

天然产物

Cat.No: T2939

Synonym: 毛喉素,Coleonol,Colforsin

Target: FXR, Adenylyl cyclase, AChR, Autophagy

Adenosine 5'-diphosphate

Cat.No: T1723

Synonym: 腺苷5'-二磷酸,Adenosine diphosphate,adenosine pyrophosphate,ADP

Target: Endogenous Metabolite

Prostaglandin E1

Cat.No: T1626

Synonym: 前列地尔,PGE1,列腺素E1,Alprostadil

Target: Endogenous Metabolite, Prostaglandin Receptor

Cat.No: T16332

Synonym: Colforsin dapropate hydrochloride

Target: NMDAR

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